Summary

Name CHRM4
Full Name Muscarinic acetylcholine receptor M4
Synonyms ACM4_HUMAN |
Primary ID P08173
Links - -
Type protein
Relations 19
Inhibitors atropine; dothiepin; Hexocyclium; amitriptyline
Function The muscarinic acetylcholine receptor mediates various cellular responses, including inhibition of adenylate cyclase, breakdown of phosphoinositides and modulation of potassium channels through the action of G proteins. Primary transducing effect is inhibition of adenylate cyclase.

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Relations

Regulator Mechanism target score
+ up-regulates activity img/direct-activation.png chemical activation CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus
+ down-regulates activity img/direct_inhibition.png chemical inhibition CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus
+ down-regulates activity img/direct_inhibition.png chemical inhibition CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png binding GNAI1 0.427
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation CHRM4 0.8
Publications: 1 Organism: Rattus Norvegicus
+ up-regulates activity img/direct-activation.png binding GNAI3 0.371
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation CHRM4 0.8
Publications: 2 Organism: Homo Sapiens, Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus
+ down-regulates activity img/direct_inhibition.png chemical inhibition CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png binding GNAO1 0.354
Publications: 1 Organism: Homo Sapiens
+ down-regulates activity img/direct_inhibition.png chemical inhibition CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation CHRM4 0.8
Publications: 1 Organism: Cricetulus Griseus