Summary

Name EDNRA
Full Name Endothelin-1 receptor
Synonyms Endothelin A receptor, ET-A, ETA-R, hET-AR | ETA, ETRA
Primary ID P25101
Links - -
Type protein
Relations 14
Inhibitors N-(3-methoxy-5-methyl-2-pyrazinyl)-2-[4-(1,3,4-oxadiazol-2-yl)phenyl]-3-pyridinesulfonamide; sitaxentan
Function Receptor for endothelin-1. Mediates its action by association with G proteins that activate a phosphatidylinositol-calcium second messenger system. The rank order of binding affinities for ET-A is

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Relations

Regulator Mechanism target score
+ up-regulates activity img/direct-activation.png chemical activation EDNRA 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAO1 0.276
Publications: 1 Organism: Homo Sapiens
+ down-regulates img/direct_inhibition.png chemical inhibition EDNRA 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAI3 0.418
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAZ 0.251
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding GNA13 0.541
Publications: 1 Organism: Homo Sapiens
Tissue: Kidney
+ up-regulates activity img/direct-activation.png binding GNAI1 0.389
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNA14 0.442
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAS 0.449
Publications: 1 Organism: Homo Sapiens
+ down-regulates activity img/direct_inhibition.png chemical inhibition EDNRA 0.8
Publications: 1 Organism: In Vitro
+ up-regulates img/direct-activation.png binding EDNRA 0.878
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAQ 0.52
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding GNAQ 0.52
Publications: 1 Organism: Homo Sapiens
Tissue: Muscle, Smooth Muscle
+ up-regulates activity img/direct-activation.png binding GNAL 0.42
Publications: 1 Organism: Homo Sapiens