| Modifier | Substrate | Residue | Sequence | Mechanism/Effect | PMID | Interaction ID |
|---|---|---|---|---|---|---|
| GRK2 | ADRA2A | Ser314 | DLEESSSsDHAERPP | phosphorylation down-regulates activity | 7876239 | SIGNOR-251443 |
| Enzyme | Effect | Phosphosite | Effect | Target | PMID | Interaction ID |
|---|---|---|---|---|---|---|
| GRK2 | phosphorylation up-regulates → | ADRA2A PSer314 | phosphorylation down-regulates ⊣ | ADRA2A | 7876239 | SIGNOR-251443 |
| Regulator | Mechanism/Effect | Target | SIGNOR-ID |
|---|---|---|---|
| GRK2 | phosphorylation → down-regulates activity | ADRA2A | SIGNOR-251443 |