| Modifier | Substrate | Residue | Sequence | Mechanism/Effect | PMID | Interaction ID |
|---|---|---|---|---|---|---|
| SRC | AR | Tyr535 | MDSYSGPyGDMRLET | phosphorylation up-regulates activity | 20383201 | SIGNOR-278168 |
| EPHA3 | AR | Tyr535 | MDSYSGPyGDMRLET | phosphorylation up-regulates activity | 20570899 | SIGNOR-279370 |
| Enzyme | Effect | Phosphosite | Effect | Target | PMID | Interaction ID |
|---|---|---|---|---|---|---|
| SRC | phosphorylation up-regulates → | AR PTyr535 | phosphorylation up-regulates → | AR | 20383201 | SIGNOR-278168 |
| EPHA3 | phosphorylation up-regulates → | AR PTyr535 | phosphorylation up-regulates → | AR | 20570899 | SIGNOR-279370 |
| Regulator | Mechanism/Effect | Target | SIGNOR-ID |
|---|---|---|---|
| SRC | phosphorylation → up-regulates activity | AR | SIGNOR-278168 |
| EPHA3 | phosphorylation → up-regulates activity | AR | SIGNOR-279370 |