| Name | KIT |
| ID | P10721 |
| Role | kinase |
| Enzymatic Domains |
Ig-like C2-type 1 27-112
Ig-like C2-type 2 121-205
Ig-like C2-type 3 212-308
Ig-like C2-type 4 317-410
Ig-like C2-type 5 413-507
Protein kinase 589-937 PROSITE-ProRule |
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| Modifier | Substrate | Residue | Sequence | Mechanism/Effect | PMID | Interaction ID |
|---|---|---|---|---|---|---|
| KIT | KIT | Tyr703 | DHAEAALyKNLLHSK | phosphorylation up-regulates | 10377264 | SIGNOR-68643 |
| KIT | KIT | Tyr936 | SESTNHIySNLANCS | phosphorylation up-regulates | 10377264 | SIGNOR-68647 |
| KIT | KIT | Tyr568 | EEINGNNyVYIDPTQ | phosphorylation up-regulates activity | 12824176 | SIGNOR-102633 |
| KIT | KIT | Tyr570 | INGNNYVyIDPTQLP | phosphorylation up-regulates activity | 12824176 | SIGNOR-102637 |
| KIT | KIT | Tyr823 | DIKNDSNyVVKGNAR | phosphorylation up-regulates activity | 12824176 | SIGNOR-102641 |
| KIT | CBL | – | phosphorylation up-regulates activity | 15315962 | SIGNOR-279199 | |
| KIT | CTNNB1 | – | phosphorylation up-regulates activity | 17949810 | SIGNOR-278361 | |
| KIT | PHB | Tyr259 | SRSRNITyLPAGQSV | phosphorylation up-regulates activity | 32169072 | SIGNOR-278362 |
| KIT | STAT1 | Tyr701 | DGPKGTGyIKTELIS | phosphorylation up-regulates activity | 21135090 | SIGNOR-251365 |
| KIT | PTPN11 | – | phosphorylation up-regulates activity | 22806893 | SIGNOR-256140 | |
| KIT | SLA | Tyr120 | SETKKGFySLSVRHR | phosphorylation down-regulates activity | 24284075 | SIGNOR-263140 |
| KIT | SLA | Tyr258 | KKSISLMyGGSKRKS | phosphorylation down-regulates activity | 24284075 | SIGNOR-263141 |
| KIT | SLA | Tyr273 | SFFSSPPyFED | phosphorylation down-regulates activity | 24284075 | SIGNOR-263142 |
| KIT | STAP1 | – | phosphorylation up-regulates activity | 10679268 | SIGNOR-261820 | |
| KIT | PI3K | – | phosphorylation up-regulates activity | 15526160 | SIGNOR-254949 | |
| KIT | SRC_kinase_family | – | phosphorylation up-regulates | 15526160 | SIGNOR-254995 |
| Enzyme | Effect | Phosphosite | Effect | Target | PMID | Interaction ID |
|---|---|---|---|---|---|---|
| KIT | phosphorylation up-regulates → | KIT PTyr703 | phosphorylation up-regulates → | KIT | 10377264 | SIGNOR-68643 |
| KIT | phosphorylation up-regulates → | KIT PTyr936 | phosphorylation up-regulates → | KIT | 10377264 | SIGNOR-68647 |
| KIT | phosphorylation up-regulates → | KIT PTyr568 | phosphorylation up-regulates → | KIT | 12824176 | SIGNOR-102633 |
| KIT | phosphorylation up-regulates → | KIT PTyr570 | phosphorylation up-regulates → | KIT | 12824176 | SIGNOR-102637 |
| KIT | phosphorylation up-regulates → | KIT PTyr823 | phosphorylation up-regulates → | KIT | 12824176 | SIGNOR-102641 |
| KIT | phosphorylation up-regulates → | PHB PTyr259 | phosphorylation up-regulates → | PHB | 32169072 | SIGNOR-278362 |
| KIT | phosphorylation up-regulates → | STAT1 PTyr701 | phosphorylation up-regulates → | STAT1 | 21135090 | SIGNOR-251365 |
| KIT | phosphorylation up-regulates → | SLA PTyr120 | phosphorylation down-regulates ⊣ | SLA | 24284075 | SIGNOR-263140 |
| KIT | phosphorylation up-regulates → | SLA PTyr258 | phosphorylation down-regulates ⊣ | SLA | 24284075 | SIGNOR-263141 |
| KIT | phosphorylation up-regulates → | SLA PTyr273 | phosphorylation down-regulates ⊣ | SLA | 24284075 | SIGNOR-263142 |
| Regulator | Mechanism/Effect | Target | SIGNOR-ID |
|---|---|---|---|
| KIT | phosphorylation → up-regulates | KIT | SIGNOR-68643 |
| KIT | phosphorylation → up-regulates | KIT | SIGNOR-68647 |
| KIT | phosphorylation → up-regulates activity | KIT | SIGNOR-102633 |
| KIT | phosphorylation → up-regulates activity | KIT | SIGNOR-102637 |
| KIT | phosphorylation → up-regulates activity | KIT | SIGNOR-102641 |
| KIT | phosphorylation → up-regulates activity | CBL | SIGNOR-279199 |
| KIT | phosphorylation → up-regulates activity | CTNNB1 | SIGNOR-278361 |
| KIT | phosphorylation → up-regulates activity | PHB | SIGNOR-278362 |
| KIT | phosphorylation → up-regulates activity | STAT1 | SIGNOR-251365 |
| KIT | phosphorylation → up-regulates activity | PTPN11 | SIGNOR-256140 |
| KIT | phosphorylation → down-regulates activity | SLA | SIGNOR-263140 |
| KIT | phosphorylation → down-regulates activity | SLA | SIGNOR-263141 |
| KIT | phosphorylation → down-regulates activity | SLA | SIGNOR-263142 |
| KIT | phosphorylation → up-regulates activity | STAP1 | SIGNOR-261820 |
| KIT | phosphorylation → up-regulates activity | PI3K | SIGNOR-254949 |
| KIT | phosphorylation → up-regulates | SRC_kinase_family | SIGNOR-254995 |