| Modifier | Substrate | Residue | Sequence | Mechanism/Effect | PMID | Interaction ID |
|---|---|---|---|---|---|---|
| PRKCG | GRK2 | Ser29 | ATPAARAsKKILLPE | phosphorylation up-regulates activity | 11042191 | SIGNOR-249060 |
| PRKCD | GRK2 | Ser29 | ATPAARAsKKILLPE | phosphorylation up-regulates activity | 11042191 | SIGNOR-249059 |
| PRKCA | GRK2 | Ser29 | ATPAARAsKKILLPE | phosphorylation up-regulates activity | 11042191 | SIGNOR-249058 |
| PRKCG | GRK2 | Ser29 | ATPAARAsKKILLPE | phosphorylation up-regulates | 11042191 | SIGNOR-83231 |
| Enzyme | Effect | Phosphosite | Effect | Target | PMID | Interaction ID |
|---|---|---|---|---|---|---|
| PRKCG | phosphorylation up-regulates → | GRK2 PSer29 | phosphorylation up-regulates → | GRK2 | 11042191 | SIGNOR-249060 |
| PRKCD | phosphorylation up-regulates → | GRK2 PSer29 | phosphorylation up-regulates → | GRK2 | 11042191 | SIGNOR-249059 |
| PRKCA | phosphorylation up-regulates → | GRK2 PSer29 | phosphorylation up-regulates → | GRK2 | 11042191 | SIGNOR-249058 |
| PRKCG | phosphorylation up-regulates → | GRK2 PSer29 | phosphorylation up-regulates → | GRK2 | 11042191 | SIGNOR-83231 |
| Regulator | Mechanism/Effect | Target | SIGNOR-ID |
|---|---|---|---|
| PRKCG | phosphorylation → up-regulates activity | GRK2 | SIGNOR-249060 |
| PRKCD | phosphorylation → up-regulates activity | GRK2 | SIGNOR-249059 |
| PRKCA | phosphorylation → up-regulates activity | GRK2 | SIGNOR-249058 |
| PRKCG | phosphorylation → up-regulates | GRK2 | SIGNOR-83231 |