Summary

Name AVPR2
Full Name Vasopressin V2 receptor
Synonyms V2R, AVPR V2, Antidiuretic hormone receptor, Renal-type arginine vasopressin receptor | ADHR, DIR, DIR3, V2R
Primary ID P30518
Links - -
Type protein
Relations 5
Inhibitors conivaptan
Function Receptor for arginine vasopressin. The activity of this receptor is mediated by G proteins which activate adenylate cyclase. Involved in renal water reabsorption.

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Relations

Regulator Mechanism target score
+ up-regulates activity img/direct-activation.png binding GNAS 0.565
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation AVPR2 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding AVPR2 0.728
Publications: 1 Organism: Homo Sapiens
Tissue: Muscle, Kidney, Smooth Muscle
+ up-regulates activity img/direct-activation.png binding GNAL 0.272
Publications: 1 Organism: Homo Sapiens
+ down-regulates activity img/direct_inhibition.png chemical inhibition AVPR2 0.8
Publications: 1 Organism: In Vitro