| + |
CID 132010322 | down-regulates activity
chemical inhibition
|
BRD4 |
0.8 |
| Identifier |
Residue |
Sequence |
Organism |
Cell Line |
| SIGNOR-261102 |
|
|
Homo sapiens |
|
| pmid |
sentence |
| 31969702 |
ABBV-744 potently inhibited the BD2 domain of BET family proteins with more than 290× selectivity relative to the BD1 domains of BRD2, BRD3 and BRD4 |
|
| Publications: |
1 |
Organism: |
Homo Sapiens |
| + |
CID 132010322 | down-regulates activity
chemical inhibition
|
BRD2 |
0.8 |
| Identifier |
Residue |
Sequence |
Organism |
Cell Line |
| SIGNOR-261103 |
|
|
Homo sapiens |
|
| pmid |
sentence |
| 31969702 |
ABBV-744 potently inhibited the BD2 domain of BET family proteins with more than 290× selectivity relative to the BD1 domains of BRD2, BRD3 and BRD4 |
|
| Publications: |
1 |
Organism: |
Homo Sapiens |
| + |
CID 132010322 | down-regulates activity
chemical inhibition
|
BRD3 |
0.8 |
| Identifier |
Residue |
Sequence |
Organism |
Cell Line |
| SIGNOR-261104 |
|
|
Homo sapiens |
|
| pmid |
sentence |
| 31969702 |
ABBV-744 potently inhibited the BD2 domain of BET family proteins with more than 290× selectivity relative to the BD1 domains of BRD2, BRD3 and BRD4 |
|
| Publications: |
1 |
Organism: |
Homo Sapiens |