Summary

Name MC5R
Full Name Melanocortin receptor 5
Synonyms MC5-R, MC-2
Primary ID P33032
Links - -
Type protein
Relations 17
Function Receptor for MSH (alpha, beta and gamma) and ACTH. The activity of this receptor is mediated by G proteins which activate adenylate cyclase. This receptor is a possible mediator of the immunomodulation properties of melanocortins.

Viewer

Relations

Regulator Mechanism target score
+ up-regulates img/direct-activation.png binding MC5R 0.762
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNA14 0.27
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAL 0.295
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding MC5R 0.762
Publications: 1 Organism: Homo Sapiens
Tissue: Brain
+ up-regulates activity img/direct-activation.png binding GNAS 0.444
Publications: 2 Organism: Homo Sapiens
+ down-regulates activity img/direct_inhibition.png binding MC5R 0.511
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png binding GNAZ 0.251
Publications: 1 Organism: Homo Sapiens
+ down-regulates activity img/direct_inhibition.png binding MC5R 0.509
Publications: 1 Organism: Homo Sapiens
Tissue: Brain
+ down-regulates activity img/direct_inhibition.png binding MC5R 0.402
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png binding GNAI1 0.251
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAQ 0.251
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNA12 0.251
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAI3 0.251
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding MC5R 0.2
Publications: 1 Organism: Homo Sapiens
Tissue: Brain
+ up-regulates activity img/direct-activation.png chemical activation MC5R 0.8
Publications: 1 Organism: Homo Sapiens
+ down-regulates activity img/direct_inhibition.png binding MC5R 0.561
Publications: 1 Organism: Homo Sapiens
Tissue: Brain