Summary

Name CDK16
Full Name Cyclin-dependent kinase 16
Synonyms Cell division protein kinase 16, PCTAIRE-motif protein kinase 1, Serine/threonine-protein kinase PCTAIRE-1 | PCTAIRE1, PCTK1
Primary ID Q00536
Links - -
Type protein
Relations 7
Inhibitors dabrafenib
Function Protein kinase that plays a role in vesicle-mediated transport processes and exocytosis. Regulates GH1 release by brain neurons. Phosphorylates NSF, and thereby regulates NSF oligomerization. Required for normal spermatogenesis. Regulates neuron differentiation and dendrite development (By similarity). Plays a role in the regulation of insulin secretion in response to changes in blood glucose levels. Can phosphorylate CCNY at 'Ser-336' (in vitro).

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Modifications Tables

Relations

Regulator Mechanism target score
+ down-regulates quantity by destabilization img/direct_inhibition.png phosphorylation CDKN1B 0.339
Publications: 1 Organism: Homo Sapiens
+ down-regulates img/direct_inhibition.png phosphorylation CDK16 0.32
Publications: 1 Organism: Homo Sapiens
Tissue: Brain
+ up-regulates activity img/direct-activation.png phosphorylation CDK16 0.688
Publications: 1
+ up-regulates activity img/direct-activation.png phosphorylation PRKAR1A 0.275
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png phosphorylation PRC1 0.351
Publications: 1 Organism: Homo Sapiens
+ form complex img/form-complex.png binding CyclinY/CDK16 0.688
Publications: 1
+ down-regulates activity img/direct_inhibition.png chemical inhibition CDK16 0.8
Publications: 1 Organism: Homo Sapiens