Summary

Name PTGER1
Full Name Prostaglandin E2 receptor EP1 subtype
Synonyms PGE receptor EP1 subtype, PGE2 receptor EP1 subtype, Prostanoid EP1 receptor
Primary ID P34995
Links - -
Type protein
Relations 8
Function Receptor for prostaglandin E2 (PGE2). The activity of this receptor is mediated by G(q) proteins which activate a phosphatidylinositol-calcium second messenger system. May play a role as an important modulator of renal function. Implicated the smooth muscle contractile response to PGE2 in various tissues.

Viewer

Relations

Regulator Mechanism target score
+ up-regulates activity img/direct-activation.png binding GNA14 0.403
Publications: 1 Organism: Homo Sapiens
+ down-regulates quantity by repression img/indirect_inhibition.png transcriptional regulation PTGER1 0.2
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNA12 0.265
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation PTGER1 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAS 0.427
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding GNAQ 0.419
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAL 0.251
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAQ 0.419
Publications: 1 Organism: Homo Sapiens