Summary
| Name | LY-2157299
|
| Synonyms | galunisertib (WHO MedNet), galunisertib (WHO MedNet), galunisertib (WHO MedNet), galunisertibum (WHO MedNet), LY 2157299 (SUBMITTER), LY2157299 (SUBMITTER) |
| IUPAC | 4-[2-(6-methylpyridin-2-yl)-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazol-3-yl]quinoline-6-carboxamide |
| Formula | C22H19N5O |
| PRIMARY ID (Read more) |
CHEBI:137064![]() |
| Type | chemical |
| Relations | 3 |
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Relations
| Regulator | Mechanism | target | score ℹ | |
|---|---|---|---|---|
| + | LY-2157299 | down-regulates
chemical inhibition
|
TGFBR1 | 0.8 |
| Publications: | 2 | Organism: | Homo Sapiens | |
| + | LY-2157299 | down-regulates
chemical inhibition
|
TGFBR2 | 0.8 |
| Publications: | 1 | Organism: | Homo Sapiens | |
4.0
LY-2157299

chemical inhibition