Summary

Name ADRA2C
Full Name Alpha-2C adrenergic receptor
Synonyms Alpha-2 adrenergic receptor subtype C4, Alpha-2C adrenoreceptor, Alpha-2C adrenoceptor, Alpha-2CAR | ADRA2L2, ADRA2RL2
Primary ID P18825
Links - -
Type protein
Relations 17
Inhibitors tolazoline; lurasidone
Function Alpha-2 adrenergic receptors mediate the catecholamine-induced inhibition of adenylate cyclase through the action of G proteins.

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Relations

Regulator Mechanism target score
+ up-regulates activity img/direct-activation.png chemical activation ADRA2C 0.8
Publications: 1 Organism: In Vitro
+ up-regulates activity img/direct-activation.png binding GNAZ 0.406
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation ADRA2C 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation ADRA2C 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAO1 0.404
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation ADRA2C 0.8
Publications: 2 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation ADRA2C 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation ADRA2C 0.8
Publications: 1 Organism: Homo Sapiens
+ down-regulates activity img/direct_inhibition.png chemical inhibition ADRA2C 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation ADRA2C 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation ADRA2C 0.8
Publications: 1 Organism: Homo Sapiens
+ down-regulates activity img/direct_inhibition.png chemical inhibition ADRA2C 0.8
Publications: 1 Organism: Cricetulus Longicaudatus
+ up-regulates activity img/direct-activation.png binding GNAI1 0.452
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAI3 0.461
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation ADRA2C 0.8
Publications: 1 Organism: Cricetulus Longicaudatus
+ up-regulates activity img/direct-activation.png chemical activation ADRA2C 0.8
Publications: 1 Organism: Homo Sapiens