Summary

Name LPAR3
Full Name Lysophosphatidic acid receptor 3
Synonyms LPA receptor 3, LPA-3, Lysophosphatidic acid receptor Edg-7 | EDG7, LPA3
Primary ID Q9UBY5
Links - -
Type protein
Relations 19
Inhibitors 3-[({4-[4-({[1-(2-chlorophenyl)ethoxy]carbonyl}amino)-3-methyl-1,2-oxazol-5-yl]phenyl}methyl)sulfanyl]propanoic acid
Function Receptor for lysophosphatidic acid (LPA), a mediator of diverse cellular activities. May play a role in the development of ovarian cancer. Seems to be coupled to the G(i)/G(o) and G(q) families of heteromeric G proteins.

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Relations

Regulator Mechanism target score
+ up-regulates activity img/direct-activation.png binding GNAI1 0.429
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding GNA13 0.382
Publications: 2 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding GNA12 0.438
Publications: 2 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNA14 0.474
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAL 0.251
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNA15 0.405
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAI3 0.432
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png chemical activation LPAR3 0.8
Publications: 3 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding GNAQ 0.456
Publications: 1 Organism: Homo Sapiens
+ down-regulates img/direct_inhibition.png chemical inhibition LPAR3 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding GNAI1 0.429
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAO1 0.251
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAQ 0.456
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation LPAR3 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAZ 0.251
Publications: 1 Organism: Homo Sapiens