Summary

Name GPR17
Full Name Uracil nucleotide/cysteinyl leukotriene receptor
Synonyms UDP/CysLT receptor, G-protein coupled receptor 17, P2Y-like receptor, R12 |
Primary ID Q13304
Links - -
Type protein
Relations 5
Function Dual specificity receptor for uracil nucleotides and cysteinyl leukotrienes (CysLTs). Signals through G(i) and inhibition of adenylyl cyclase. May mediate brain damage by nucleotides and CysLTs following ischemia.

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Relations

Regulator Mechanism target score
+ up-regulates activity img/direct-activation.png binding GNAO1 0.2
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAI1 0.38
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAQ 0.352
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAI3 0.354
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation GPR17 0.8
Publications: 1 Organism: Homo Sapiens