Summary

Name DRD3
Full Name D
Synonyms Dopamine D3 receptor |
Primary ID P35462
Links - -
Type protein
Relations 34
Pathways Dopaminergic Synapse
Inhibitors 2-[4-[3-[2-(trifluoromethyl)-9-thioxanthenylidene]propyl]-1-piperazinyl]ethanol; pimozide; (S)-(-)-sulpiride; cis-(z)-Flupenthixol; chlorpromazine; sulpiride; amisulpride; 3-phenanthryl hydrogen sulfate; sertindole; domperidone; zotepine; haloperidol; LSM-20934; clozapine
Function Dopamine receptor whose activity is mediated by G proteins which inhibit adenylyl cyclase. Promotes cell proliferation.

Viewer

Relations

Regulator Mechanism target score
+ up-regulates activity img/direct-activation.png chemical activation DRD3 0.8
Publications: 1 Organism: In Vitro
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 1 Organism: Cricetulus Griseus
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 2 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation DRD3 0.8
Publications: 1 Organism: In Vitro
+ up-regulates activity img/direct-activation.png chemical activation DRD3 0.8
Publications: 3 Organism: Cricetulus Griseus, Homo Sapiens
Pathways:Dopaminergic Synapse
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 1 Organism: Cricetulus Griseus
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation DRD3 0.8
Publications: 2 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation DRD3 0.8
Publications: 1 Organism: In Vitro
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 1 Organism: Cricetulus Griseus
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 1 Organism: In Vitro
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 1 Organism: Cricetulus Griseus
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 1 Organism: In Vitro
+ up-regulates activity img/direct-activation.png binding GNAI1 0.547
Publications: 1 Organism: Homo Sapiens
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 1 Organism: Chlorocebus Aethiops
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 2 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png binding GNAZ 0.316
Publications: 1 Organism: Homo Sapiens
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 1 Organism: Chlorocebus Aethiops
+ up-regulates activity img/direct-activation.png binding GNAO1 0.464
Publications: 1 Organism: Homo Sapiens
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation DRD3 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png binding GNB5 0.451
Publications: 1 Organism: Homo Sapiens
Pathways:Dopaminergic Synapse
+ up-regulates activity img/direct-activation.png chemical activation DRD3 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation DRD3 0.8
Publications: 1 Organism: In Vitro
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png binding GNAI3 0.454
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation DRD3 0.8
Publications: 1 Organism: In Vitro
+ down-regulates activity img/direct_inhibition.png chemical inhibition DRD3 0.8
Publications: 1 Organism: Cricetulus Griseus
+ up-regulates activity img/direct-activation.png chemical activation DRD3 0.8
Publications: 1 Organism: Cricetulus Griseus