Summary

Name CCKBR
Full Name Gastrin/cholecystokinin type B receptor
Synonyms CCK-B receptor, CCK-BR, Cholecystokinin-2 receptor, CCK2-R | CCKRB
Primary ID P32239
Links - -
Type protein
Relations 11
Function Receptor for gastrin and cholecystokinin. The CCK-B receptors occur throughout the central nervous system where they modulate anxiety, analgesia, arousal, and neuroleptic activity. This receptor mediates its action by association with G proteins that activate a phosphatidylinositol-calcium second messenger system.; FUNCTION

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Relations

Regulator Mechanism target score
+ up-regulates activity img/direct-activation.png binding GNAL 0.268
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAQ 0.424
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation CCKBR 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAS 0.267
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding CCKBR 0.867
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNA15 0.483
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAO1 0.256
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAI3 0.27
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding CCKBR 0.777
Publications: 1 Organism: Homo Sapiens
Tissue: Brain
+ up-regulates activity img/direct-activation.png binding GNAI1 0.277
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNA14 0.423
Publications: 1 Organism: Homo Sapiens