Summary

Name LPAR2
Full Name Lysophosphatidic acid receptor 2
Synonyms LPA receptor 2, LPA-2, Lysophosphatidic acid receptor Edg-4 | EDG4, LPA2
Primary ID Q9HBW0
Links - -
Type protein
Relations 16
Inhibitors 3-[({4-[4-({[1-(2-chlorophenyl)ethoxy]carbonyl}amino)-3-methyl-1,2-oxazol-5-yl]phenyl}methyl)sulfanyl]propanoic acid
Function Receptor for lysophosphatidic acid (LPA), a mediator of diverse cellular activities. Seems to be coupled to the G(i)/G(o), G(12)/G(13), and G(q) families of heteromeric G proteins. Plays a key role in phospholipase C-beta (PLC-beta) signaling pathway. Stimulates phospholipase C (PLC) activity in a manner that is independent of RALA activation.

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Relations

Regulator Mechanism target score
+ down-regulates img/direct_inhibition.png chemical inhibition LPAR2 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding GNA13 0.384
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding GNAI1 0.609
Publications: 2 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png chemical activation LPAR2 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAI1 0.609
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAZ 0.251
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAI3 0.44
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png chemical activation LPAR2 0.8
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAQ 0.579
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAL 0.251
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAO1 0.251
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNAS 0.369
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding GNA12 0.465
Publications: 1 Organism: Homo Sapiens
+ up-regulates img/direct-activation.png binding LPAR2 0.301
Publications: 1 Organism: Homo Sapiens
+ up-regulates activity img/direct-activation.png binding GNA14 0.456
Publications: 1 Organism: Homo Sapiens